Affinity DataKi: 22nMAssay Description:Inhibitory activity against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibitory activity against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Inhibitory activity against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibitory activity against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of dopamine-sensitive rat brain adenylyl cyclase activity assessed as cAMP levelMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of dopamine-sensitive rat brain adenylyl cyclase activity assessed as cAMP levelMore data for this Ligand-Target Pair
TargetAdenylate cyclase type 1/Adenylate cyclase type 2/Adenylate cyclase type 3/Adenylate cyclase type 4/Adenylate cyclase type 5/Adenylate cyclase type 6/Adenylate cyclase type 8/Adenylyl cyclase 7(Rattus norvegicus)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:The compound was tested for adenylate cyclase activity in rat corpus striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory concentration against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibitory concentration against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
TargetAdenylate cyclase type 1/Adenylate cyclase type 2/Adenylate cyclase type 3/Adenylate cyclase type 4/Adenylate cyclase type 5/Adenylate cyclase type 6/Adenylate cyclase type 8/Adenylyl cyclase 7(Rattus norvegicus)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory concentration against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of dopamine-sensitive rat brain adenylyl cyclase activity assessed as cAMP levelMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibitory concentration against Dopamine sensitive adenylate cyclase in ratsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+3nMAssay Description:Inhibition of Rap1A-mediated geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Inhibition of Rap1A-mediated geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Inhibition of Rap1A-mediated geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair