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Found 143 of affinity data for UniProtKB/TrEMBL: O35491
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50239782(CHEMBL4082113)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant GST-tagged mouse CLK2 using GRSRSRSRSRSR as substrate after 30 mins in presence of [gamma-32P]-ATP by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259415(CHEMBL4061526)
Affinity DataIC50:  28nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594790(CHEMBL5200518)
Affinity DataIC50:  30nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259570(CHEMBL4102871)
Affinity DataIC50:  30nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259477(CHEMBL4071322)
Affinity DataIC50:  32nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594796(CHEMBL5179655)
Affinity DataIC50:  35nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259467(CHEMBL4070189)
Affinity DataIC50:  47nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259589(CHEMBL4065432)
Affinity DataIC50:  52nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50097868(CHEMBL3589661)
Affinity DataIC50:  55nMAssay Description:Inhibition of mouse recombinant CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259335(CHEMBL4072506)
Affinity DataIC50:  59nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50097867(CHEMBL3589660)
Affinity DataIC50:  61nMAssay Description:Inhibition of mouse recombinant CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594797(CHEMBL5195216)
Affinity DataIC50:  67nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50347746(CHEMBL1803085)
Affinity DataIC50:  83nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50097855(CHEMBL3589666)
Affinity DataIC50:  110nMAssay Description:Inhibition of mouse recombinant CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594773(CHEMBL5206143)
Affinity DataIC50:  110nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594765(CHEMBL5208980)
Affinity DataIC50:  120nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594771(CHEMBL5181355)
Affinity DataIC50:  120nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594785(CHEMBL5181008)
Affinity DataIC50:  120nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594784(CHEMBL5196066)
Affinity DataIC50:  130nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataIC50:  130nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50469189(CHEMBL4284209)
Affinity DataIC50:  130nMAssay Description:Inhibition of recombinant GST-tagged mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of [gamma-33P] ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259405(CHEMBL4077159)
Affinity DataIC50:  130nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259569(CHEMBL4074499)
Affinity DataIC50:  130nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594768(CHEMBL5195122)
Affinity DataIC50:  140nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259571(CHEMBL4084919)
Affinity DataIC50:  160nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259527(CHEMBL4070227)
Affinity DataIC50:  160nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594769(CHEMBL5199422)
Affinity DataIC50:  170nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259416(CHEMBL4089652)
Affinity DataIC50:  180nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594775(CHEMBL5203292)
Affinity DataIC50:  180nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50097870(CHEMBL3589664)
Affinity DataIC50:  180nMAssay Description:Inhibition of mouse recombinant CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594788(CHEMBL5179457)
Affinity DataIC50:  180nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259561(CHEMBL4092673)
Affinity DataIC50:  180nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  200nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK2 expressed in Escherichia coli DH5[alpha] using NH2-RSPSYGRSRSRSRSRSRSRSRSNSRSRSY-OH as substrate by l...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  200nMAssay Description:Inhibition of mouse Clk2Checked by AuthorMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50026622(CHEMBL408982)
Affinity DataIC50:  200nMAssay Description:Inhibition of mouse glutathione S-transferase-tagged Clk2 expressed in Escherichia coli DH5alpha using NH2-RSPSYGRSRSRSRSRSRSRSRSNSRSRSY-OH peptide a...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50443638(CHEMBL3092863)
Affinity DataIC50:  210nMAssay Description:Inhibition of mouse recombinant CLK2 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259413(CHEMBL4105084)
Affinity DataIC50:  220nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259526(CHEMBL4093104)
Affinity DataIC50:  220nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594782(CHEMBL5206744)
Affinity DataIC50:  220nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259354(CHEMBL4090223)
Affinity DataIC50:  220nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594799(CHEMBL5187753)
Affinity DataIC50:  250nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594783(CHEMBL5180765)
Affinity DataIC50:  260nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50443639(CHEMBL3092862)
Affinity DataIC50:  280nMAssay Description:Inhibition of mouse recombinant CLK2 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  280nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK2 expressed in Escherichia coli using GRSRSRSRSRSR as substrate and [gamma33P]ATP after 30 mins by scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50594774(CHEMBL5194491)
Affinity DataIC50:  320nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50347750(CHEMBL1802358)
Affinity DataIC50:  320nMAssay Description:Inhibition of mouse recombinant CLK2 expressed in Escherichia coli using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50347743(CHEMBL1803082)
Affinity DataIC50:  380nMAssay Description:Inhibition of mouse recombinant GST-fused CLK2 expressed in Escherichia coli using GRSRSRSRSRSR peptide as substrate incubated for 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259411(CHEMBL4086402)
Affinity DataIC50:  380nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50259409(CHEMBL4062820)
Affinity DataIC50:  380nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mus musculus)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50097854(CHEMBL3589665)
Affinity DataIC50:  390nMAssay Description:Inhibition of mouse recombinant CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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