Affinity DataKi: 21nMpH: 7.4Assay Description:The compound was tested for inhibition of rat plasma renin at pH of 7.4.More data for this Ligand-Target Pair
Affinity DataKi: 115nMpH: 6.0Assay Description:The compound was tested for inhibition of rat plasma renin at pH of 6.0.More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Binding affinity against nicotinic acetylcholine receptor alpha4-beta4 using [3H]epibatidine as radioligand expressed in HEK293 cells or tsA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 230nMpH: 7.4Assay Description:Inhibition of rhizopuspepsinMore data for this Ligand-Target Pair
Affinity DataKi: 630nMpH: 7.4Assay Description:Binding affinity against nicotinic acetylcholine receptor using [3H]epibatidine as radioligand in rat brain tissueMore data for this Ligand-Target Pair
Affinity DataKi: 630nMpH: 7.4Assay Description:Inhibition of rhizopuspepsinMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Inhibitory activity of the compound against renin was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.580nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound was tested for its inhibitory activity against Rat plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:In vitro inhibitory activity towards porcine kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:In vitro inhibitory activity against man (human) plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of dog plasma renin activityMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:In vitro inhibitory activity against hog plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:In vitro inhibitory activity towards porcine kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:In vitro inhibitory activity against hog plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:In vitro inhibitory activity against rat plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibitory activity of compound against renin was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:In vitro inhibitory activity against hog plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:In vitro inhibitory activity against hog plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of rat reninMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Inhibition of renin in rat plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:In vitro inhibitory activity towards porcine kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of hog man plasma renin activityMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:In vitro inhibitory activity against rat plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 199nMAssay Description:Compound was evaluated for inhibition of plasma renin activity in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of renin in rat plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair