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Found 5 of affinity data for UniProtKB/TrEMBL: P19332
TargetMicrotubule-associated protein tau(Rattus norvegicus)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50313696(CHEMBL1086427 | N-(6-chloro-7-fluoro-5-phenyl-1H-i...)
Affinity DataIC50:  250nMAssay Description:Inhibition of Tau phosphorylation in rat cerebral cortex after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Rattus norvegicus)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50313661(CHEMBL1095040 | N-(6-chloro-5-phenyl-1H-indazol-3-...)
Affinity DataIC50:  400nMAssay Description:Inhibition of Tau phosphorylation in rat cerebral cortex after 120 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein tau(Rattus norvegicus)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50487729(CHEMBL454948)
Affinity DataEC50:  2.90E+3nMAssay Description:Inhibition of microtubule polymerisation in Rattus norvegicus (rat) A10 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetMicrotubule-associated protein tau(Rattus norvegicus)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50487730(CHEMBL508222)
Affinity DataEC50:  4.40E+3nMAssay Description:Inhibition of microtubule polymerisation in Rattus norvegicus (rat) A10 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetMicrotubule-associated protein tau(Rattus norvegicus)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50340902((4-amino-2-(pyridin-3-ylamino)thiazol-5-yl)(2-fluo...)
Affinity DataEC50:  5.50E+3nMAssay Description:Inhibition of tau protein phosphorylation at Ser396 in rat brain cells at 0.5 to 50 uM after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed