Compile Data Set for Download or QSAR
maximum 50k data
Found 347 of affinity data for UniProtKB/TrEMBL: P31651
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50419338(CHEMBL1446457)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of mouse BGT1 expressed in hamster BHK cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50039251((R)-1-(4,4-bis(3-methylthiophen-2-yl)but-3-enyl)pi...)
Affinity DataIC50:  180nMAssay Description:Inhibition of [3H]GABA uptake at GAT2 in mouse astrocytes after 3 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50039251((R)-1-(4,4-bis(3-methylthiophen-2-yl)but-3-enyl)pi...)
Affinity DataIC50:  360nMAssay Description:Inhibition of [3H]GABA uptake at GAT2 in mouse neurons after 3 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50419338(CHEMBL1446457)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of mouse mGAT2 expressed in HEK293 cells assessed as inhibition of [3H]GABA uptake after 3 mins incubation by TopCount microplate scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50343258(4-((4,4-bis(3-methylthiophen-2-yl)but-3-enyl)(meth...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of [3H]GABA uptake at GAT2 in mouse astrocytes after 3 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50343258(4-((4,4-bis(3-methylthiophen-2-yl)but-3-enyl)(meth...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of [3H]GABA uptake at GAT2 in mouse neurons after 3 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50563998(CHEMBL4781266)
Affinity DataIC50:  4.47E+3nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577077(CHEMBL4854996)
Affinity DataIC50:  4.57E+3nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577076(CHEMBL4858459)
Affinity DataIC50:  5.75E+3nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021387(CHEMBL3289585)
Affinity DataIC50:  5.89E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021385(CHEMBL3289583)
Affinity DataIC50:  5.89E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021360(CHEMBL3289575)
Affinity DataIC50:  6.46E+3nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021360(CHEMBL3289575)
Affinity DataIC50:  6.46E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577069(CHEMBL4863244)
Affinity DataIC50:  6.76E+3nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021372(CHEMBL3289296)
Affinity DataIC50:  6.92E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577075(CHEMBL4856428)
Affinity DataIC50:  7.76E+3nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021377(CHEMBL3289570)
Affinity DataIC50:  7.76E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021371(CHEMBL3289295)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021390(CHEMBL3289588)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021375(CHEMBL3289568)
Affinity DataIC50:  8.91E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577073(CHEMBL4862980)
Affinity DataIC50:  9.12E+3nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021389(CHEMBL3289587)
Affinity DataIC50:  9.33E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021373(CHEMBL3289566)
Affinity DataIC50:  9.55E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021376(CHEMBL3289569)
Affinity DataIC50:  9.55E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021363(CHEMBL3289578)
Affinity DataIC50:  9.55E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577078(CHEMBL4854550)
Affinity DataIC50:  9.55E+3nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577072(CHEMBL4851621)
Affinity DataIC50:  9.77E+3nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021388(CHEMBL3289586)
Affinity DataIC50:  9.77E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021361(CHEMBL3289576)
Affinity DataIC50:  9.77E+3nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021382(CHEMBL3289580)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577071(CHEMBL4870735)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021384(CHEMBL3289582)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021383(CHEMBL3289581)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250277(CHEMBL4104932)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human BGT1/human GAT3 chimera B expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577080(CHEMBL4873878)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577074(CHEMBL4866914)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250277(CHEMBL4104932)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of mouse BGT1 expressed in HEK293 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577082(CHEMBL4861574)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021379(CHEMBL3289572)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577081(CHEMBL4852705)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021381(CHEMBL3289574)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021374(CHEMBL3289567)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021386(CHEMBL3289584)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50492898(CHEMBL2414176)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50210524(CHEMBL3941169)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptake preincubated for 25 mins followed by [3H]GABA addition mea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021362(CHEMBL3289577)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577079(CHEMBL4859850)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50021380(CHEMBL3289573)
Affinity DataIC50:  1.41E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK293 cells assessed as decrease in [3H]GABA uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577070(CHEMBL4850155)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent betaine transporter(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50577068(CHEMBL4849048)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of mouse GAT2 expressed in human HEK293 cell line assessed as inhibition of [3H]GABA uptake measured after 40 mins by LC-ESI-MS/MS analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 347 total ) | Next | Last >>
Jump to: