Compile Data Set for Download or QSAR
maximum 50k data
Found 186 for UniProtKB: P43143
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50263130((+)-7-Methyl-2-exo-[3'-(2-fluoropyridin-3-yl)-5'-p...)
Affinity DataKi:  0.0210nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50263095((+)-7-Methyl-2-exo-[3'-(2-fluoropyridin-4-yl)-5'-p...)
Affinity DataKi:  0.0310nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50263171((+)-2-(6'-[18F]fluoro-3,3'-bipyridin-5-yl)-7-methy...)
Affinity DataKi:  0.0470nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50263131((+)-7-Methyl-2-exo-[3'-(6-fluoropyridin-2-yl)-5'-p...)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50045045(CHEMBL3341965)
Affinity DataKi: >300nMAssay Description:Partial agonist activity at rat alpha6 nAChRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50334463(1,3,5-tri-{5-[1-(3-picolinium)]-pent-1-ynyl}benzen...)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-3(Rattus norvegicus)
Hainan University

Curated by ChEMBL
LigandPNGBDBM50445330(CHEMBL3104243)
Affinity DataIC50:  0.260nMAssay Description:Inhibition of rat alpha6/alpha3beta2beta3 nAChR expressed in Xenopus oocytes assessed as inhibition of ACh-induced current by voltage clamp electroph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50334472(1,3,5-tris(5-(3,4-dihydroisoquinolin-2(1H)-yl)pent...)
Affinity DataIC50:  0.350nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567433(CHEMBL4869892)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50334464(1,12-bis(3-methyl-5,6-dihydropyridin-1(2H)-yl)dode...)
Affinity DataIC50:  0.950nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50238606(CHEMBL4099865)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current at -70 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50445330(CHEMBL3104243)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus oocytes assessed as inhibition of ACh-induced current by voltage clamp electrophysiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567430(CHEMBL4860756)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567432(CHEMBL4876825)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50119774(1,1'-(dodecane-1,12-diyl)bis(3-methylpyridinium)br...)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50119774(1,1'-(dodecane-1,12-diyl)bis(3-methylpyridinium)br...)
Affinity DataIC50:  2nMAssay Description:Antagonist activity at nAChRalpha6beta2 in Sprague-Dawley rat striatal slices assessed as inhibition of nicotine-evoked [3H]dopamine uptake by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567431(CHEMBL4878931)
Affinity DataIC50:  3nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50334474(1,1',1'',1'''-(5,5',5'',5'''-(benzene-1,2,4,5-tetr...)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567435(CHEMBL4872191)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of rat alpha6/alpha3beta2beta3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50334466(1,3,5-tris(5-(3-methyl-5,6-dihydropyridin-1(2H)-yl...)
Affinity DataIC50:  3.22nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50459664(CHEMBL4218406)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50334470(1,12-bis(3,4-dihydroisoquinolin-2(1H)-yl)dodecane ...)
Affinity DataIC50:  8.59nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50547502(CHEMBL4793300)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of rat alpha6alpha3beta2beta3 expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced channel current response...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50334471(1,10-bis(3,4-dihydroisoquinolin-2(1H)-yl)decane | ...)
Affinity DataIC50:  9.91nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50459654(CHEMBL4206157)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50445326(CHEMBL3104239)
Affinity DataIC50:  11nMAssay Description:Inhibition of rat alpha6/alpha3beta2beta3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50516340(CHEMBL4439678)
Affinity DataIC50:  13nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567426(CHEMBL4878856)
Affinity DataIC50:  15nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50516340(CHEMBL4439678)
Affinity DataIC50:  17nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50516316(CHEMBL4454928)
Affinity DataIC50:  18nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50459656(CHEMBL4214931)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567413(CHEMBL4865365)
Affinity DataIC50:  21nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50459653(CHEMBL4211045)
Affinity DataIC50:  21nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567426(CHEMBL4878856)
Affinity DataIC50:  23nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50459661(CHEMBL4215453)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567413(CHEMBL4865365)
Affinity DataIC50:  27nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-3(Rattus norvegicus)
Hainan University

Curated by ChEMBL
LigandPNGBDBM50445322(CHEMBL3104235)
Affinity DataIC50:  28nMAssay Description:Inhibition of rat alpha6/alpha3beta2beta3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of ACh-induced current by voltage clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50238616(CHEMBL3104238)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 6...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50334475(3,3',3'',3'''-(1,1',1'',1'''-(5,5',5'',5'''-(benze...)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM86240(Alpha-Conotoxin MII | Gly-L-Cys(1)-L-Cys(2)-L-Ser-...)
Affinity DataIC50:  32nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50445331(CHEMBL3104245)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nAChR nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetyl choline-induced membra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50238610(CHEMBL4062759)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50334465(1,10-bis(3-methyl-5,6-dihydropyridin-1(2H)-yl)deca...)
Affinity DataIC50:  37.4nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50238580(CHEMBL4099451)
Affinity DataIC50:  39nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50238589(CHEMBL4061135)
Affinity DataIC50:  39nMAssay Description:Inhibition of noradrenaline uptake in rat synaptosomal fractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50119805(1,12-di(2-isoquinoliniumyl)dodecane; with dibromid...)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at alpha6 nAChR in rat striatum assessed as inhibition of nicotine-induced [3H]dopamine releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50238579(CHEMBL4070842)
Affinity DataIC50:  41nMAssay Description:Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567438(CHEMBL4865866)
Affinity DataIC50:  44nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567438(CHEMBL4865866)
Affinity DataIC50:  44nMAssay Description:Inhibition of rat alpha6/alpha3beta2beta3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567427(CHEMBL4872474)
Affinity DataIC50:  45nMAssay Description:Inhibition of rat alpha6/alpha3beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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