Compile Data Set for Download or QSAR
maximum 50k data
Found 63 of affinity data for UniProtKB/TrEMBL: Q01279
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50038202(5-((2,5-dihydroxybenzyl)(2-hydroxybenzyl)amino)-2-...)
Affinity DataIC50:  11.5nMAssay Description:Inhibition of mouse EGFR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50025605(CHEMBL483830)
Affinity DataIC50:  27.7nMAssay Description:Inhibition of mouse EGFR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM3294(4-Anilinoquinazoline deriv. 45 | 4-N-(3-bromopheny...)
Affinity DataIC50:  40nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50038199(5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-benzoic ac...)
Affinity DataIC50:  43.6nMAssay Description:Inhibition of mouse EGFR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50133373(CHEMBL137617 | N-(3-bromophenyl)-6-[(1E)-3-methylt...)
Affinity DataIC50:  70nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)
Affinity DataIC50:  81nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM3532(CHEMBL540068 | CHEMBL7917 | N-(3-chlorophenyl)-6,7...)
Affinity DataIC50: <100nMAssay Description:Inhibition of EGF-dependent mouse keratinocyte MK cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50136231(((2E)-3-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-...)
Affinity DataIC50:  110nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50136228(((2E)-3-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-...)
Affinity DataIC50:  130nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50505838(CHEMBL4537790)
Affinity DataIC50:  190nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50133371(CHEMBL137189 | N-(3-methylphenyl)-6-[(1E)-3-methyl...)
Affinity DataIC50:  200nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50505845(CHEMBL4566193)
Affinity DataIC50:  270nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50025591(CHEMBL483831)
Affinity DataIC50:  445nMAssay Description:Inhibition of mouse EGFR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50136230(6-[(1E)-3-acetyl-3-methyltriaz-1-enyl]-N-(3-methyl...)
Affinity DataIC50:  578nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50505841(CHEMBL4532034 | US11174245, # I-018)
Affinity DataIC50:  700nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  750nMAssay Description:Inhibition of mouse EGFR by liquid scintillation countingMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50102422(5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-(3-pheny...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of epidermal growth factor receptor phosphorylation in BaF3 mouse lymphoid cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50505846(CHEMBL4562138)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM3973(N-[(E)-2-(2,5-dihydroxyphenyl)ethenyl]formamide | ...)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of mouse EGFR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50505842(CHEMBL4519157)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50025606(LAVENDUSTIN B)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of mouse EGFR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50505840(CHEMBL4550104)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50478479(CHEMBL520491)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of mouse EGFR by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50074740(3-(3-Chloro-phenyl)-5-hydroxy-7-methoxy-1-methyl-1...)
Affinity DataIC50:  2.83E+3nMAssay Description:Inhibition of EGF-dependent mouse keratinocyte MK cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50505843(CHEMBL4449589 | US11174245, # I-235)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50102416(5-(2,5-Dihydroxy-benzylamino)-N-[2-(4-fluoro-pheny...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of epidermal growth factor receptor phosphorylation in BaF3 mouse lymphoid cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50102415(5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-(1,2,3,4...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of epidermal growth factor receptor phosphorylation in BaF3 mouse lymphoid cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50074739(3-(3-Chloro-phenyl)-5-hydroxy-7-methoxy-1-phenethy...)
Affinity DataIC50:  4.93E+3nMAssay Description:Inhibition of EGF-dependent mouse keratinocyte MK cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50505839(CHEMBL4525935 | US11174245, # I-001)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50102421(CHEMBL140774 | N-Benzyl-5-(2,5-dihydroxy-benzylami...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of epidermal growth factor receptor phosphorylation in BaF3 mouse lymphoid cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50074742(CHEMBL7866 | [3-(3-Chloro-phenyl)-5-hydroxy-7-meth...)
Affinity DataIC50:  9.55E+3nMAssay Description:Inhibition of EGF-dependent mouse keratinocyte MK cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50162993(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Epidermal growth factor receptor in P19 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50162996(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Epidermal growth factor receptor in P19 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50162990(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Epidermal growth factor receptor in P19 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50162994(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Epidermal growth factor receptor in P19 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50162991(3-(1-Benzo[b]thiophen-2-yl-1H-indol-3-yl)-4-[1-(3-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Epidermal growth factor receptor in P19 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50102423(5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-phenethy...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of epidermal growth factor receptor phosphorylation in BaF3 mouse lymphoid cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Epidermal growth factor receptor in P19 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50162998(3-[1-(3-Dimethylamino-propyl)-1H-indazol-3-yl]-4-(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Epidermal growth factor receptor in P19 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50505836(CHEMBL4434788 | US11174245, # I-064)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of wild type EGFR in mouse BAF3 cells assessed as reduction in cell proliferation incubated for 72 hrs by Celltiter-Glo luminescent cell v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50074743(3-(3-Chloro-phenyl)-5,7-dihydroxy-1H-quinolin-4-on...)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of EGF-dependent mouse keratinocyte MK cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50066984(4-(5-(4-hydroxybenzyl)-4-(4-methoxybenzyl)-1-methy...)
Affinity DataIC50:  1.13E+4nMAssay Description:Inhibition of Epidermal growth factor receptor mediated mitogenesis of NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50074744(3-(3-Chloro-phenyl)-5-hydroxy-7-methoxy-1H-quinoli...)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of EGF-dependent mouse keratinocyte MK cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50102414(5-(2,5-Dihydroxy-benzylamino)-N-hexyl-2-hydroxy-be...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of epidermal growth factor receptor phosphorylation in BaF3 mouse lymphoid cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50102427(5-(2,5-Dihydroxy-benzylamino)-2-hydroxy-N-(2-pyrid...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of epidermal growth factor receptor phosphorylation in BaF3 mouse lymphoid cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50074745(3-(3-Chloro-phenyl)-5,7-dihydroxy-chromen-4-one | ...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of EGF-dependent mouse keratinocyte MK cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM60918(5-Amino-2-hydroxy-benzoic acid | MESALAMINE | MLS0...)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of mouse EGFR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50066983(5-[1-(4-Hydroxy-benzyl)-4-(4-methoxy-benzyl)-1H-im...)
Affinity DataIC50:  2.27E+4nMAssay Description:Inhibition of Epidermal growth factor receptor mediated mitogenesis of NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50102418(4-(2,5-Dihydroxy-benzylamino)-N-(3-phenyl-propyl)-...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of epidermal growth factor receptor phosphorylation in BaF3 mouse lymphoid cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Mus musculus)TBA
LigandPNGBDBM50102420(5-(2,5-Dihydroxy-benzylamino)-N-dodecyl-2-hydroxy-...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of epidermal growth factor receptor phosphorylation in BaF3 mouse lymphoid cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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