Affinity DataIC50: 3.60nMAssay Description:Displacement of [125I]human ghrelin from rat GHS-R1a expressed in HEK cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of rat HDAC1 using Boc-Lys(Ac)-AMC as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.55E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 3.01E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 3.03E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 3.18E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 3.19E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of HDAC1 in rat liver extract by trypsin assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 7.53E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Rattus norvegicus)
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Chengdu University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 8.76E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair