Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of affinity data for UniProtKB/TrEMBL: Q5RLM2
TargetSolute carrier family 22 member 7(Rattus norvegicus)
Kyorin University

Curated by ChEMBL
LigandPNGBDBM20688((3R,5R)-7-[(1S,2S,6S,8S,8aR)-6-hydroxy-2-methyl-8-...)
Affinity DataIC50:  4.49E+5nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha uptake (PGF2: 50nM) in rOAT2-expressing S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 7(Rattus norvegicus)
Kyorin University

Curated by ChEMBL
LigandPNGBDBM50206509(4-Dipropylsulfamoyl-benzoic acid | 4-Dipropylsulfa...)
Affinity DataIC50:  9.77E+5nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha uptake (PGF2: 50nM) in rOAT2-expressing S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 7(Rattus norvegicus)
Kyorin University

Curated by ChEMBL
LigandPNGBDBM82898((6R,7R)-3-(acetoxymethyl)-8-keto-7-[[2-(2-thienyl)...)
Affinity DataIC50:  1.50E+6nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha in OAT2-S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 7(Rattus norvegicus)
Kyorin University

Curated by ChEMBL
LigandPNGBDBM50390999(CEFOPERAZONE)
Affinity DataIC50:  1.62E+6nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha in OAT2-S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 7(Rattus norvegicus)
Kyorin University

Curated by ChEMBL
LigandPNGBDBM50350468(CEFAMANDOLE)
Affinity DataIC50:  3.18E+6nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha in OAT2-S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 7(Rattus norvegicus)
Kyorin University

Curated by ChEMBL
LigandPNGBDBM50350473(Aliporina | CEFALORIDINE)
Affinity DataIC50: >5.00E+6nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha in OAT2-S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 7(Rattus norvegicus)
Kyorin University

Curated by ChEMBL
LigandPNGBDBM50335523((6R,7R)-3-(acetoxymethyl)-7-(2-(2-aminothiazol-4-y...)
Affinity DataIC50: >5.00E+6nMAssay Description:TP_TRANSPORTER: inhibition of PGF2alpha in OAT2-S2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed