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Found 108 of affinity data for UniProtKB/TrEMBL: Q61606
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566470(CHEMBL4857523)
Affinity DataIC50:  0.530nMAssay Description:Antagonist activity at mouse GCGR expressed in CHO-K1 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50566469(CHEMBL4876736)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at mouse GCGR expressed in CHO-K1 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075766(4-[5-(4-Chloro-phenyl)-3-(2-propoxy-phenyl)-1H-pyr...)
Affinity DataIC50:  30nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075775(4-[3-(5-Bromo-2-propoxy-phenyl)-5-(4-chloro-phenyl...)
Affinity DataIC50:  37nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075787(4-[3-(4-Bromo-2-propoxy-phenyl)-5-(4-chloro-phenyl...)
Affinity DataIC50:  49nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the human glucagon receptor (GGR) expressed on CH...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075783(4-[5-(4-Chloro-phenyl)-3-(5-chloro-2-propoxy-pheny...)
Affinity DataIC50:  50nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075780(4-[5-(4-Chloro-phenyl)-3-isopropyl-1H-pyrrol-2-yl]...)
Affinity DataIC50:  60nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075748(4-[5-(4-Chloro-phenyl)-3-cyclohexyl-1H-pyrrol-2-yl...)
Affinity DataIC50:  60nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075772(4-[3-(2-Butoxy-phenyl)-5-(4-chloro-phenyl)-1H-pyrr...)
Affinity DataIC50:  80nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007239(CHEMBL3238226)
Affinity DataIC50:  84nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007231(CHEMBL3238221)
Affinity DataIC50:  90nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007240(CHEMBL3238228)
Affinity DataIC50:  96nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007228(CHEMBL3238219)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007223(CHEMBL3238215)
Affinity DataIC50:  110nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007219(CHEMBL3238214)
Affinity DataIC50:  110nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50360601(CHEMBL1933349 | MK-0893)
Affinity DataIC50:  122nMAssay Description:Antagonist activity at mouse GCGR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation preincubated for 30 mins prior ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007226(CHEMBL3238218)
Affinity DataIC50:  130nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007296(CHEMBL3238246)
Affinity DataIC50:  130nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007225(CHEMBL3238217)
Affinity DataIC50:  140nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007233(CHEMBL3238223)
Affinity DataIC50:  140nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075752(4-[5-(4-Chloro-phenyl)-3-(2-isobutoxy-phenyl)-1H-p...)
Affinity DataIC50:  150nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007224(CHEMBL3238216)
Affinity DataIC50:  160nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007232(CHEMBL3238222)
Affinity DataIC50:  170nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007230(CHEMBL3238220)
Affinity DataIC50:  190nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007241(CHEMBL3238229)
Affinity DataIC50:  200nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50071899(4-[5-(4-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrr...)
Affinity DataIC50:  200nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075764(4-[3,5-Bis-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyrid...)
Affinity DataIC50:  220nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075751(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-...)
Affinity DataIC50:  230nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075767(4-[3-(3-Bromo-phenyl)-5-(4-chloro-phenyl)-1H-pyrro...)
Affinity DataIC50:  230nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075758(4-[5-(4-Chloro-phenyl)-3-(4-methoxy-phenyl)-1H-pyr...)
Affinity DataIC50:  240nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075775(4-[3-(5-Bromo-2-propoxy-phenyl)-5-(4-chloro-phenyl...)
Affinity DataIC50:  250nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075749(4-[3-(2-Allyloxy-phenyl)-5-(4-chloro-phenyl)-1H-py...)
Affinity DataIC50:  270nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007218(CHEMBL3237928)
Affinity DataIC50:  280nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007214(CHEMBL3237925)
Affinity DataIC50:  310nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075754(4-[5-(4-Chloro-phenyl)-3-(2-ethoxy-phenyl)-1H-pyrr...)
Affinity DataIC50:  340nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075757(4-[5-(2,4-Dichloro-phenyl)-3-(4-fluoro-phenyl)-1H-...)
Affinity DataIC50:  340nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075784(4-[5-(4-Chloro-phenyl)-3-(2-hexyloxy-phenyl)-1H-py...)
Affinity DataIC50:  340nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007210(CHEMBL3237922)
Affinity DataIC50:  370nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075786(4-[5-(4-Chloro-phenyl)-3-(2-methoxy-phenyl)-1H-pyr...)
Affinity DataIC50:  400nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007440(CHEMBL3237917)
Affinity DataIC50:  400nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007212(CHEMBL3237924)
Affinity DataIC50:  420nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007215(CHEMBL3237927)
Affinity DataIC50:  420nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075753(4-[3,5-Bis-(4-fluoro-phenyl)-1H-pyrrol-2-yl]-pyrid...)
Affinity DataIC50:  430nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075781(CHEMBL348555 | {2-[5-(4-Chloro-phenyl)-2-pyridin-4...)
Affinity DataIC50:  440nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the human glucagon receptor (GGR) expressed on CH...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075788(4-[5-(3-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrr...)
Affinity DataIC50:  460nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007211(CHEMBL3237923)
Affinity DataIC50:  500nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075750(5-(4-Chloro-phenyl)-2-pyridin-4-yl-1H-pyrrole-3-ca...)
Affinity DataIC50:  500nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50007245(CHEMBL3238234)
Affinity DataIC50:  520nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075763(4-[5-(4-Chloro-phenyl)-3-(2,6-dipropoxy-phenyl)-1H...)
Affinity DataIC50:  670nMAssay Description:Binding affinity determined by reduction in binding of 125 I-glucagon to the human glucagon receptor expressed on CHO cells in absence of Mg+2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50075766(4-[5-(4-Chloro-phenyl)-3-(2-propoxy-phenyl)-1H-pyr...)
Affinity DataIC50:  700nMAssay Description:Binding affinity determined by reduction in binding of 125 I-glucagon to the human glucagon receptor expressed on CHO cells in absence of Mg+2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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