Compile Data Set for Download or QSAR
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Found 3 of affinity data for UniProtKB/TrEMBL: Q80T02
TargetG-protein coupled bile acid receptor 1(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50428095(CHEMBL2331646)
Affinity DataEC50:  3.93E+3nMAssay Description:Agonist activity at rat TGR5 expressed in deoxycycline-induced CHO cells assessed as increase in intracellular cAMP measured after 48 hrs by HTRF com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50414955(CHEMBL576138)
Affinity DataEC50:  631nMAssay Description:Agonist activity at rat TGR5 expressed in melanophores assessed as melanosome dispersion by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetG-protein coupled bile acid receptor 1(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50414954(CHEMBL575966)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at rat TGR5 expressed in melanophores assessed as melanosome dispersion by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed