Affinity DataEC50: 3.93E+3nMAssay Description:Agonist activity at rat TGR5 expressed in deoxycycline-induced CHO cells assessed as increase in intracellular cAMP measured after 48 hrs by HTRF com...More data for this Ligand-Target Pair
Affinity DataEC50: 631nMAssay Description:Agonist activity at rat TGR5 expressed in melanophores assessed as melanosome dispersion by melanophore assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Agonist activity at rat TGR5 expressed in melanophores assessed as melanosome dispersion by melanophore assayMore data for this Ligand-Target Pair