Compile Data Set for Download or QSAR
maximum 50k data
Found 70 of affinity data for UniProtKB/TrEMBL: Q8NCG7
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50532885(CHEMBL4470017)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of human GST-tagged DAGLbeta catalytic domain expressed in HEK293F cell membranes using EnzChek as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50532885(CHEMBL4470017)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of human GST-tagged DAGLbeta catalytic domain expressed in HEK293F cell membranes using EnzChek as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50532882(CHEMBL4476210)
Affinity DataIC50:  25nMAssay Description:Inhibition of human GST-tagged DAGLbeta catalytic domain expressed in HEK293F cell membranes using EnzChek as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50532882(CHEMBL4476210)
Affinity DataIC50:  25nMAssay Description:Inhibition of human GST-tagged DAGLbeta catalytic domain expressed in HEK293F cell membranes using EnzChek as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50147615(CHEMBL3764876)
Affinity DataIC50:  40nMAssay Description:Inhibition of DAGLbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50148158(CHEMBL3764017)
Affinity DataIC50:  40nMAssay Description:Inhibition of DAGLbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM24567((2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant DAGLbeta overexpressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50240877(CHEMBL158897 | Quinolyl derivatives | cyclohexanon...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant DAGLbeta overexpressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50148187(CHEMBL3764093)
Affinity DataIC50:  80nMAssay Description:Inhibition of DAGLbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50147618(CHEMBL3765022)
Affinity DataIC50:  112nMAssay Description:Inhibition of DAGLbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50147617(CHEMBL3765421)
Affinity DataIC50:  146nMAssay Description:Inhibition of DAGLbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50211257(CHEMBL3895863 | US10583137, Compound 14)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434939(N-(2-ethylbutyl)-N-(2-(pyridin- 3-yl)ethyl)-4-(4- ...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434937(N-neopentyl-N-(2-(pyridin-3- yl)ethyl)-4-(4- (trif...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434935(N-neopentyl-N-(2-(pyridin-4- yl)ethyl)-4-(4- (trif...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434933(N-(cyclopropylmethyl)-N- phenethyl-4-(4- (trifluor...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434930(N-neopentyl-N-phenethyl-4-(4- (trifluoromethoxy)ph...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434929(N-(2-ethylbutyl)-N-phenethyl-4- (4-(trifluorometho...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434928(N-cyclopropyl-N-phenethyl-4- (4-(trifluoromethoxy)...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434927(N-cyclobutyl-N-phenethyl-4-(4- (trifluoromethoxy)p...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434926(N-neopentyl-N-phenethyl-4-(4- (trifluoromethoxy)ph...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434925(N-(2-ethylbutyl)-N-phenethyl-4- (4-(trifluorometho...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434920((2-benzylpiperidin-1-yl)(4-(6- bromopyridin-3-yl)-...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434919((2-benzylpiperidin-1-yl)(4-(4- nitrophenyl)-1H-1,2...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434918(4-(1-(2-benzylpiperidine-1- carbonyl)-1H-1,2,3-tri...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434913((2-benzylpiperidin-1-yl)(4-(4- methoxyphenyl)-1H-1...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434908((2-benzylpiperidin-1-yl)(4-(4- (4,6-dimethoxypyrim...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434908((2-benzylpiperidin-1-yl)(4-(4- (4,6-dimethoxypyrim...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434899((2-benzylpiperidin-1-yl)(4-(4- (3,5-dichloropyridi...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434892((4-([1,1'-biphenyl]-4-yl)-1H- 1,2,3-triazol-1-yl)(...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434882(N-(2-Ethylbutyl)-N-(2-(pyridin-4-yl)ethyl)-4-(4-(t...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434881((2-Benzylpiperidin-1-yl)(4-(2′,4′,6...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434880((2-Benzylpiperidin-1-yl)(4-(4-(3,5-dimethoxypyridi...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434879(US10583137, Compound 17 | tert-Butyl 3-benzyl-4-(4...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM24567((2S)-1-[(2S,3S)-3-hexyl-4-oxooxetan-2-yl]tridecan-...)
Affinity DataIC50:  420nMAssay Description:Inhibition of DAGLbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434898((2-benzylpiperidin-1-yl)(4-(4- (3,5-difluoropyridi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434924((2-benzylpiperidin-1-yl)(4-(4- (morpholinomethyl)p...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434903(4'-(1-(2-benzylpiperidine-1- carbonyl)-1H-1,2,3-tr...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434936(N-neopentyl-N-(2-(pyridin-4- yl)ethyl)-4-(4- (trif...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434932(N-cyclopropyl-N-phenethyl-4- (4-(trifluoromethoxy)...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434940(US10583137, Compound 137)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434934(N-(cyclopropylmethyl)-N- phenethyl-4-(4- (trifluor...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434880((2-Benzylpiperidin-1-yl)(4-(4-(3,5-dimethoxypyridi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434931(N-cyclobutyl-N-phenethyl-4-(4- (trifluoromethoxy)p...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434893((2-(pyridin-4- ylmethyl)piperidin-1-yl)(4- (2',4',...)
Affinity DataIC50:  6.00E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434922((2-benzylpiperidin-1-yl)(4-(4- ((dimethylamino)met...)
Affinity DataIC50:  6.00E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434891((2-benzylpiperidin-1-yl)(4-(4-(3- methoxypyridin-4...)
Affinity DataIC50:  6.00E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434890((2-benzylpiperidin-1-yl)(4-(2',6'- dimethoxy-4'-me...)
Affinity DataIC50:  6.00E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434889((2-benzylpiperidin-1-yl)(4-(2',6'- dimethoxy-[1,1'...)
Affinity DataIC50:  6.00E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM434887((2-benzylpiperidin-1-yl)(4-(2',4'- dimethoxy-[1,1'...)
Affinity DataIC50:  6.00E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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