Compile Data Set for Download or QSAR
maximum 50k data
Found 100 of affinity data for UniProtKB/TrEMBL: Q8TDS5
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50210259((4Z,7Z,10Z,13Z,16Z,19Z)-docosa-4,7,10,13,16,19-hex...)
Affinity DataKi:  1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50269534((8Z,11Z,14Z)-Icosatrienoic acid | (8Z,11Z,14Z)-ico...)
Affinity DataKi:  3.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50242349((5Z,8Z,11Z,14Z,17Z)-5,8,11,14,17-eicosapentaenoic ...)
Affinity DataKi:  6.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465693(CHEMBL4283608)
Affinity DataIC50:  0.120nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465682(CHEMBL4287941)
Affinity DataIC50:  0.280nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465685(CHEMBL4281149)
Affinity DataIC50:  0.380nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465690(CHEMBL4282356)
Affinity DataIC50:  2.10nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50054792(CHEMBL3341973)
Affinity DataIC50:  2.20nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50054794(CHEMBL3341971)
Affinity DataIC50:  2.70nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50024458(5-oxo-ETE | CHEMBL18028 | ETE-5-Oxo)
Affinity DataIC50:  3nMAssay Description:Desensitization of 5-oxo-ETE receptor in indo-1-labeled human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50054793(CHEMBL3341972)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446952(CHEMBL3115775)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50054793(CHEMBL3341972)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50054793(CHEMBL3341972)
Affinity DataIC50:  6nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446953(CHEMBL3115774)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446953(CHEMBL3115774)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50341133((6E,8Z,11Z,14Z)-20,20,20-trifluoro-5-oxoicosa-6,8,...)
Affinity DataIC50:  7.5nMAssay Description:Desensitization of 5-oxo-ETE receptor in indo-1-labeled human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465692(CHEMBL4284672)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465681(CHEMBL4277299)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446952(CHEMBL3115775)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446953(CHEMBL3115774)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446952(CHEMBL3115775)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446953(CHEMBL3115774)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at 5-oxo-ETE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced Ca2+ mobilization incubated for 2 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465695(CHEMBL4291346)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50262197(CHEMBL4084871)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465684(CHEMBL4291464)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446954(CHEMBL3115793)
Affinity DataIC50:  26nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446953(CHEMBL3115774)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in anti-CD49d-labeled eosinophils assessed as inhibition of 5-oxo-ETE-induced F-actin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446961(CHEMBL3115786)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446952(CHEMBL3115775)
Affinity DataIC50:  33nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in anti-CD49d-labeled eosinophils assessed as inhibition of 5-oxo-ETE-induced F-actin ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465680(CHEMBL4278772)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465683(CHEMBL4279605)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446955(CHEMBL3115792)
Affinity DataIC50:  81nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446965(CHEMBL3115782)
Affinity DataIC50:  90nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465686(CHEMBL4277207)
Affinity DataIC50:  120nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446964(CHEMBL3115783)
Affinity DataIC50:  136nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446962(CHEMBL3115785)
Affinity DataIC50:  141nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465691(CHEMBL4280693)
Affinity DataIC50:  210nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465688(CHEMBL4287509)
Affinity DataIC50:  223nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465689(CHEMBL4285167)
Affinity DataIC50:  260nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446956(CHEMBL3115791)
Affinity DataIC50:  314nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446960(CHEMBL3115787)
Affinity DataIC50:  323nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50431178(CHEMBL2332562)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as 5-oxo-ETE-induced Ca2+ mobilization incubated for 2 mins prior to 5-oxo-ETE addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446953(CHEMBL3115774)
Affinity DataIC50:  402nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in neutrophils assessed as inhibition of 5-oxo-ETE-induced cell migration after 2 hrs ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446952(CHEMBL3115775)
Affinity DataIC50:  454nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in neutrophils assessed as inhibition of 5-oxo-ETE-induced cell migration after 2 hrs ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50046281(CHEMBL3311230)
Affinity DataIC50:  460nMAssay Description:Antagonist activity at 5-oxo-ETE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced Ca2+ mobilization incubated for 2 mins pri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446976(CHEMBL3115777 | CHEMBL3115778)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization by spectrofluorometric anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50465687(CHEBI:34146 | CHEMBL1526258)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446969(CHEMBL3115800)
Affinity DataIC50:  550nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxoeicosanoid receptor 1(Homo sapiens (Human))
Tanabe Seiyaku

Curated by PDSP Ki Database
LigandPNGBDBM50446957(CHEMBL3115790)
Affinity DataIC50:  566nMAssay Description:Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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