TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 38.6nMAssay Description:Inhibition of human LCK2 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of ICK (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 53.3nMAssay Description:Inhibition of human LCK2 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant ICK (1 to 312 residues) using RRRFRPASPLRGP as substrate after 40 mins by [gamma-33ATP] by radiometric scintillation ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human LCK2 using MBP as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LCK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of NanoLuc-fused ICK (unknown origin) expressed in HEK293T cells after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ICKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 39nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 5.90E+3nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ICKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 470nMAssay Description:Binding affinity to ICKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ICKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ICKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to ICKMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.20E+3nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.20nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 0.690nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 680nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase ICK(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ICK kinase domainMore data for this Ligand-Target Pair