BDBM341808 US10544104, Compound 124::US9765037, Compound 124

SMILES CC(C)COc1ccc2cc(ccc2c1)-c1nn(CC2CCN(C)CC2)c2ncnc(N)c12

InChI Key InChIKey=GOKRPYKIPRDTFC-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 341808   

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Washington Through Its Center For

US Patent
LigandPNGBDBM341808(US9765037, Compound 124 | US10544104, Compound 124)
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Washington Through Its Center For

US Patent
LigandPNGBDBM341808(US9765037, Compound 124 | US10544104, Compound 124)
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of human tyrosine kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
University of Washington Through Its Center For

US Patent
LigandPNGBDBM341808(US9765037, Compound 124 | US10544104, Compound 124)
Affinity DataIC50: 7.85E+3nMAssay Description:Inhibition of TgCDPK1 and CpCDPK1 was determined using a luminescent kinase assay which measures ATP depletion in the presence of the Syntide 2 pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2020
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
University of Washington Through Its Center For

US Patent
LigandPNGBDBM341808(US9765037, Compound 124 | US10544104, Compound 124)
Affinity DataIC50: 7.85E+3nMAssay Description:Inhibition of human tyrosine kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/29/2019
Entry Details
US Patent