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BDBM15237 4-[1-(cyclopropylmethyl)-4-(4-fluorophenyl)-1H-imidazol-5-yl]pyridine::CHEMBL96741::PYRIDINYLIMIDAZOLE::SB2::SB216995

SMILES: Fc1ccc(cc1)-c1ncn(CC2CC2)c1-c1ccncc1

InChI Key: InChIKey=ROKOFZNQCIIJMI-UHFFFAOYSA-N

Data: 6 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 15237
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mitogen-activated protein kinase 14 (Human)	BDBM15237 (SB2 \| CHEMBL96741 \| 4-[1-(cyclopropylmethyl)-4-(4-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	160	n/a	n/a	n/a	n/a	7.5	37
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mitogen-activated protein kinase 1 (Rat)	BDBM15237 (SB2 \| CHEMBL96741 \| 4-[1-(cyclopropylmethyl)-4-(4-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.5	37
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mitogen-activated protein kinase 14 (Human)	BDBM15237 (SB2 \| CHEMBL96741 \| 4-[1-(cyclopropylmethyl)-4-(4-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	160	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Prostaglandin G/H synthase 1 (Sheep)	BDBM15237 (SB2 \| CHEMBL96741 \| 4-[1-(cyclopropylmethyl)-4-(4-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	5.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Polyunsaturated fatty acid 5-lipoxygenase (Rat)	BDBM15237 (SB2 \| CHEMBL96741 \| 4-[1-(cyclopropylmethyl)-4-(4-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mitogen-activated protein kinase 14 (Human)	BDBM15237 (SB2 \| CHEMBL96741 \| 4-[1-(cyclopropylmethyl)-4-(4-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	160	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair