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BDBM273241 2-(4-(2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-3-isopropyl-1H-indol-5-yl) piperidin-1-yl)acetamide::US10071079, Example 15::US10478424, Example 15::US11661431, Example A-1

SMILES: CC(C)c1c([nH]c2ccc(cc12)C1CCN(CC(N)=O)CC1)-c1cn2ncnc2c(C)c1C

InChI Key: InChIKey=SNFVHLQYHFQOEP-UHFFFAOYSA-N

Data: 7 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 273241   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Toll-like receptor 7


(Human)
BDBM273241
PNG
(2-(4-(2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridi...)
GoogleScholar
UniChem
n/an/a 1.40n/an/an/an/an/a25


TBA



Citation and Details
More data for this
Ligand-Target Pair
Toll-like receptor 8


(Human)
BDBM273241
PNG
(2-(4-(2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridi...)
GoogleScholar
UniChem
n/an/a 1.40n/an/an/an/an/a25


TBA



Citation and Details
More data for this
Ligand-Target Pair
Toll-like receptor 9


(Human)
BDBM273241
PNG
(2-(4-(2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridi...)
GoogleScholar
UniChem
n/an/a 5.11E+3n/an/an/an/an/a25


TBA



Citation and Details
More data for this
Ligand-Target Pair
Toll-like receptor 7


(Human)
BDBM273241
PNG
(2-(4-(2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridi...)
GoogleScholar
UniChem
n/an/a 1.40n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Toll-like receptor 8


(Human)
BDBM273241
PNG
(2-(4-(2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridi...)
GoogleScholar
UniChem
n/an/a 1.40n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Toll-like receptor 9


(Human)
BDBM273241
PNG
(2-(4-(2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridi...)
GoogleScholar
UniChem
n/an/a 5.11E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Multidrug and toxin extrusion protein 2


(Human)
BDBM273241
PNG
(2-(4-(2-(7,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridi...)
GoogleScholar
UniChem
n/an/a 300n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair