BindingDB PrimarySearch

BDBM31005 2-methyl-1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyrazino[1,2-a]azepine::MIANSERIN HYDROCHLORIDE::MLS000069681::SMR000058472::cid_68551

SMILES: CN1CCN2C(C1)c1ccccc1Cc1ccccc21

InChI Key: InChIKey=UEQUQVLFIPOEMF-UHFFFAOYSA-N

Data: 54 KI 35 IC50 3 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 92 hits for monomerid = 31005
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
5-hydroxytryptamine receptor 1D (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	380	n/a	n/a	n/a	n/a	n/a	n/a
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Transporter (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	22	n/a	n/a	n/a	n/a	n/a	n/a
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Sodium-dependent serotonin transporter (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	2.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-2C adrenergic receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	43	n/a	n/a	n/a	n/a	n/a	n/a
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Histamine H1 receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.40	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.55E+3	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2C (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	7.40	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-2A adrenergic receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	21	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2A (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	10	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 7 (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	115	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 1E (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	37.8	n/a	n/a	7.4	23
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Alpha-1A adrenergic receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	407	n/a	n/a	n/a	n/a	n/a	n/a
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D(4) dopamine receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.31E+3	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	7.08E+3	n/a	n/a	n/a	n/a	n/a	n/a
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D(3) dopamine receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.89E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	0.0700	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	380	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	210	n/a	n/a	n/a	n/a	n/a	n/a
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Histamine H2 receptor (Guinea pig)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	880	n/a	n/a	n/a	n/a	n/a	n/a
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Histamine H1 receptor (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	0.00600	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M5 (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Sphingosine 1-phosphate receptor 3 (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	>4.00E+4	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 1A (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	5.00E+4	n/a	n/a	7.4	23
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D(3) dopamine receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.89E+3	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 1A (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	398	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.55E+3	n/a	n/a	n/a	n/a	n/a	n/a
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D(4) dopamine receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.31E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-2C adrenergic receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	43	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2A (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	21	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	407	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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D(2) dopamine receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	7.08E+3	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 1D (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	380	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 1A (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	398	n/a	n/a	n/a	n/a	n/a	n/a
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Histamine H2 receptor (Guinea pig)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A/Alpha-2A adrenergic receptor (Bovine)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A/Alpha-2A adrenergic receptor (Bovine)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	300	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A/Alpha-2A adrenergic receptor (Bovine)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	6	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Serotonin 2 (5-HT2) receptor (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	1.10	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2C (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	1.40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Serotonin 2 (5-HT2) receptor (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	1.40	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2A (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	1.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2C (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	1.70	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Histamine H1 receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	1.70	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2A (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	2.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 6 (Mouse)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	3.24	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2A (Rat)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	3.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Alpha-2C adrenergic receptor (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	3.80	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2C (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	3.80	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 2A (Human)	BDBM31005 (MIANSERIN HYDROCHLORIDE \| SMR000058472 \| MLS000069...) Show SMILES Show InChI	GoogleScholar	UniChem	4.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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