BindingDB PrimarySearch

BDBM39341 11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one::11-[2-(4-methyl-1-piperazinyl)-1-oxoethyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one;hydrochloride::11-[2-(4-methylpiperazin-1-yl)acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one;hydrochloride::11-[2-(4-methylpiperazin-1-yl)ethanoyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one;hydrochloride::11-[2-(4-methylpiperazino)acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one;hydrochloride::CHEMBL9967::MLS000069702::PIRENZEPINE::PIRENZEPINE DIHYDROCHLORIDE::SMR000058502::cid_185248

SMILES: CN1CCN(CC(=O)N2c3ccccc3C(=O)Nc3cccnc23)CC1

InChI Key: InChIKey=RMHMFHUVIITRHF-UHFFFAOYSA-N

Data: 117 KI 91 IC50 1 Kd

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 209 hits for monomerid = 39341
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Genome polyprotein (WNV)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Bile salt export pump (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	>1.00E+6	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M3 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M2 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	800	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M2 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	120	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	119	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M2 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	690	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.80	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M3 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	300	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M2 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	968	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M5 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	341	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M3 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	956	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	28	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M4 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	247	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	22	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	19	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.5	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M4 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.05E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M4 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.05E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M4 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	49	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	21	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1 (Human)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	21	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M5 (Mouse)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	750	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	430	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	790	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	740	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	850	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	270	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	520	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	650	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	820	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	290	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	310	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	480	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
TBA				More data for this Ligand-Target Pair
Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	450	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
TBA								Citation and Details
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	900	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	1.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	710	n/a	n/a	n/a	n/a	n/a	n/a
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Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 (Rat)	BDBM39341 (PIRENZEPINE DIHYDROCHLORIDE \| SMR000058502 \| MLS00...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	900	n/a	n/a	n/a	n/a	n/a	n/a
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