Found 41 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM39341'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 120nMAssay Description:Inhibition of carbachol-induced release of alpha-amylase from pancreatic acinar cells from that of rat ileum contained the muscarinic acetylcholine r...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 174nMAssay Description:Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 251nMAssay Description:Compound was evaluated for displacement of [3H]-QNB from human Muscarinic m2 receptor in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 267nMAssay Description:Displacement of [3H]QNB (quinuclidinyl benzylate) from muscarinic M2 receptor of rat heart homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 267nMAssay Description:Displacement of [3H](-)-quinuclidinyl benzilate(QNB) from muscarinic (M2) receptor in rat heart homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 267nMAssay Description:Ability to displace [3H](-)-quinuclidinyl bezilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 270nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M2 by measuring displacement of [3H]-QNB from guinea pig heartMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 377nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 524nMAssay Description:Binding affinity to human M2 muscarinic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 610nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Inhibition of binding of [3H]N-methylscopolamine to muscarinic receptor (M2) in rat heart homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Evaluation of antagonistic affinity against muscarinic receptor (M3) in guinea pig ileumMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 1.83E+4nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:Displacement of [3H]-methylscopolamine binding to muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataIC50: 968nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M2 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity towards muscarinic receptor of gastric fundus containing Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair