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BDBM477065 US10882859, Reference compound PF-06263276

SMILES: CCc1cc(O)c(F)cc1-c1ccc2c(n[nH]c2c1)-c1nc2CCN(Cc2[nH]1)C(=O)c1cnc(cn1)N1CCCCC1

InChI Key: InChIKey=XDJGNPSZQSWJCV-UHFFFAOYSA-N

Data: 4 Kd

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 477065
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Tyrosine-protein kinase JAK1 (Human)	BDBM477065 (US10882859, Reference compound PF-06263276) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	2.70	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK2 (Human)	BDBM477065 (US10882859, Reference compound PF-06263276) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	0.780	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase JAK3 (Human)	BDBM477065 (US10882859, Reference compound PF-06263276) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.90	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Non-receptor tyrosine-protein kinase TYK2 (Human)	BDBM477065 (US10882859, Reference compound PF-06263276) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.90	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair