BDBM50118792 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID::2-(carboxyformamido)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-3-carboxylic acid::CHEMBL139393
SMILES OC(=O)C(=O)Nc1sc2CNCCc2c1C(O)=O
InChI Key InChIKey=ZIBMATWHOAGNTR-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 19 hits for monomerid = 50118792
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Inhibition of PTP1B I219A mutantMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 290nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 710nMAssay Description:Inhibition of TCPTP I220A mutantMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Inhibition of human recombinant Protein-tyrosine phosphatase 1B.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of wild type PTP1BMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 9.40E+3nMpH: 7.0Assay Description:Inhibition of T cell protein tyrosine phosphatase (TC-PTP) at pH 7.0More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Inhibition of TCPTPMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 1.15E+4nMAssay Description:Inhibition of PTP1B after 10 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataKi: 5.01E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 5.90E+4nMAssay Description:Inhibition of PTPRCMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase beta(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 5.60E+5nMAssay Description:Inhibition of PTPRBMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: 1.10E+6nMAssay Description:Inhibition of PTPREMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase alpha(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of PTPRAMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 6(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of PTPN6More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University Of Miami
Curated by ChEMBL
University Of Miami
Curated by ChEMBL
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of PTPRFMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of PTP1B after 10 minsMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of PTP1B by pNPP hydrolase assayMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Amherst College
Curated by ChEMBL
Amherst College
Curated by ChEMBL
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of PTP1B after 10 minsMore data for this Ligand-Target Pair