BDBM50374608 CHEMBL410295
SMILES CN1CCN(CC1)c1ccc(Nc2ncc3c(n2)n2c(nc4ccccc24)n(-c2c(C)cccc2C)c3=O)cc1
InChI Key InChIKey=BHJJWVDKNXABFS-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 21 hits for monomerid = 50374608
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of JNK3 by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibition of b-Raf by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK5 by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MSK1 by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human T-cell receptor zeta chain phosphorylation in Jurkat cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of Lck by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of Src by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of Lyn by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of ZAP-70 by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Tyk2 by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of JAK3 by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of Btk by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of c-Met by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of JNK2 by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of p38-alpha by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of Syk by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of Itk by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of Tie-2 by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Erk1 by HTRF assayMore data for this Ligand-Target Pair