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Found 86 with Last Name = 'morita' and Initial = 'h'
TargetSubstance-P receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50225899((+/-)-4-[(N-(2-methoxy-5-trifluoromethoxybenzyl)am...)
Affinity DataIC50:  0.220nMAssay Description:Displacement of [3H]substance P from NK1 human receptor expressed in IM9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50000041((+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-a...)
Affinity DataIC50:  0.630nMAssay Description:Displacement of [3H]substance P from NK1 human receptor expressed in IM9 cellsMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50225898((2-Methoxy-benzyl)-((2S,3S,3aR,6aS)-2-phenyl-octah...)
Affinity DataIC50:  3.40nMAssay Description:Displacement of [3H]substance P from NK1 human receptor expressed in IM9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020299((R-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-7-phenyl-h...)
Affinity DataIC50:  32nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50:  43nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50199522((+)-huperzine A | (+-)-HA | (-)-1-Amino-13-ethylid...)
Affinity DataIC50:  53nMAssay Description:Inhibition of bovine acetylcholinesteraseMore data for this Ligand-Target Pair
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50405735(CHEMBL2114230)
Affinity DataIC50:  71nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataIC50:  140nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020299((R-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-7-phenyl-h...)
Affinity DataIC50:  240nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020302((S-isomer)7-{2-[5-(4-Azido-phenyl)-3-hydroxy-pent-...)
Affinity DataIC50:  330nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020303((R-isomer)7-{2-[5-(4-Azido-3-iodo-phenyl)-3-hydrox...)
Affinity DataIC50:  350nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308527(10-methoxy-N(1)-methylburnamine-17-O-veratrate | C...)
Affinity DataIC50:  500nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50405735(CHEMBL2114230)
Affinity DataIC50:  670nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308529(CHEMBL589220 | Methyl (14E)-19-[(benzoyloxy)methyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308533(CHEMBL589254 | Methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50483304(11-Epi-Tubulysin D)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50483306(CHEBI:80036 | Tubulysin D)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50483305(13-Epi-Tubulysin D)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020301((R-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-7-phenyl-h...)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding potency towards PGF-2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes (BCLM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308528(Alstiphyllanine D | CHEMBL540945)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308532((14E)-14-ethylidene-6-methoxy-19-(methoxycarbonyl)...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308527(10-methoxy-N(1)-methylburnamine-17-O-veratrate | C...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50201171((1S,9R)-1-amino-13-[2-hydroxy-eth-(E)-ylidene]-11-...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of bovine erythrocyte acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308531((14E)-19-{[(3,4-dimethoxyphenyl)carbonyloxy]methyl...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308533(CHEMBL589254 | Methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308528(Alstiphyllanine D | CHEMBL540945)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020306((S-isomer)7-{2-[5-(4-Azido-2-hydroxy-phenyl)-3-hyd...)
Affinity DataIC50:  6.10E+3nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50483307(CHEMBL1643767)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by microtubule assembly assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020302((S-isomer)7-{2-[5-(4-Azido-phenyl)-3-hydroxy-pent-...)
Affinity DataIC50:  7.00E+3nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308530(CHEMBL602442 | Methyl (14E)-14-ethylidene-6-hydrox...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020303((R-isomer)7-{2-[5-(4-Azido-3-iodo-phenyl)-3-hydrox...)
Affinity DataIC50:  7.00E+3nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in bovine corpora lutea plasma membranes...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50201170(CHEMBL241838 | carinatumins B (2))
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of bovine erythrocyte acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50148881(Acetic acid (2S,3R)-8-hydroxy-2,3,9-trimethyl-4-ox...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of the polymerization of tubulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160802(2,4-Bis-(4-hydroxy-benzyl)-3-[2-(3-hydroxy-phenyl)...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160801(4-(4-Hydroxy-benzyl)-3-[2-(3-hydroxy-phenyl)-ethyl...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308532((14E)-14-ethylidene-6-methoxy-19-(methoxycarbonyl)...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50020305((R-isomer)7-{2-[4-(3-Azido-5-hydroxy-phenoxy)-3-hy...)
Affinity DataIC50:  1.10E+4nMAssay Description:Binding potency towards Prostaglandin F2 alpha receptor (competitive binding) with natural [3H]-PGF 2 alpha in ovine luteal cells (OLC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308535(CHEMBL601712 | methyl (14E)-14-ethylidene-6-methox...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT2 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50308529(CHEMBL589220 | Methyl (14E)-19-[(benzoyloxy)methyl...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of alpha-D-[U-14C]glucopyranoside uptake at human SGLT1 expressed in african green monkey COS1 cells after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50316419(CHEMBL1097908 | Gneyulin B)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of SGLT2 transfected in african green monkey COS1 cells assessed as alpha-D-[U-14C]glucopyranoside uptake after 30 mins by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50223709(CHEMBL240094 | cryptadine B)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of bovine acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50271482(CHEMBL455781 | lycoparin C)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of acetylcholinesterase from bovine erythrocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50316418(CHEMBL1097907 | Gneyulin A)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of SGLT2 transfected in african green monkey COS1 cells assessed as alpha-D-[U-14C]glucopyranoside uptake after 30 mins by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Hoshi University

Curated by ChEMBL
LigandPNGBDBM50316418(CHEMBL1097907 | Gneyulin A)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of SGLT1 transfected in african green monkey COS1 cells assessed as alpha-D-[U-14C]glucopyranoside uptake after 30 mins by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160804(4,4''-Dimethoxy-[1,1'']biphenanthrenyl-2,7,2'',7''...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160803(4,4''-Dimethoxy-9,10,9'',10''-tetrahydro-[1,3'']bi...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160805(1-(4-Hydroxy-benzyl)-4,8-dimethoxy-phenanthrene-2,...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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