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Found 60 with Last Name = 'payá' and Initial = 'm'
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50115777((E)-1-(4'-Fluorophenyl)-3-(3'',4'',5''-trimethoxyp...)
Affinity DataIC50:  30nMAssay Description:Inhibitory concentration of the compound required to produce 50% inhibition of the response was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50269843(Bolinaquinone | CHEMBL477692)
Affinity DataIC50:  100nMAssay Description:Inhibition of bee venom group 3 secretory phospholipase A2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50269843(Bolinaquinone | CHEMBL477692)
Affinity DataIC50:  200nMAssay Description:Inhibition of human synovial recombinant group 2 secretory phospholipase A2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50115783(3-(5-Ethoxy-2,4-dimethoxy-phenyl)-1-(2-trifluorome...)
Affinity DataIC50:  280nMAssay Description:Inhibitory concentration of the compound required to produce 50% inhibition of the response was determined; range-0.150.47 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Università

Curated by ChEMBL
LigandPNGBDBM50269843(Bolinaquinone | CHEMBL477692)
Affinity DataIC50:  400nMAssay Description:Inhibition of pig pancreatic group 1 secretory phospholipase A2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50066343(5-Hydroxy-4-[6-hydroxy-5-((2E,6E)-3,7,11-trimethyl...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity against bee secretory Phospholipase A2 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50259941(CHEMBL470339 | Petrosaspongiolide M)
Affinity DataIC50:  600nMAssay Description:Inhibition of bee venom secretory PLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50115779(1-(2,4-Difluoro-phenyl)-3-(5-ethoxy-2,4-dimethoxy-...)
Affinity DataIC50:  640nMAssay Description:Inhibitory concentration of the compound required to produce 50% inhibition of the response was determined; range-0.431.12 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50115780(3-(2,4-Dimethoxy-phenyl)-1-(2-trifluoromethyl-phen...)
Affinity DataIC50:  840nMAssay Description:Inhibitory concentration of the compound required to produce 50% inhibition of the response was determined; range-0.461.81 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50066343(5-Hydroxy-4-[6-hydroxy-5-((2E,6E)-3,7,11-trimethyl...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity against human synovial recombinant Phospholipase enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50115778(3-(2,5-Dimethoxy-phenyl)-1-(2-trifluoromethyl-phen...)
Affinity DataIC50:  910nMAssay Description:Inhibitory concentration of the compound required to produce 50% inhibition of the response was determined; range-0.431.85 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50115781((E)-1-(2-(trifluoromethyl)phenyl)-3-(2,4,6-trimeth...)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibitory concentration of the compound required to produce 50% inhibition of the response was determined; range-0.811.70 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50259952(CHEMBL480874 | cacospongionolide E)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human synovial group2 sPLA2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-alkyl-2-acetylglycerophosphocholine esterase(Sus scrofa)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085497(2-(ethylamino)hexadecan-1-ol | 2-Ethylamino-hexade...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of secretory PLA2 activity in porcine pancreas using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50259941(CHEMBL470339 | Petrosaspongiolide M)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human synovial secretory PLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50066342(5-Hydroxy-4-[5-((2E,6E)-3,7,11-trimethyl-dodeca-2,...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory activity against bee secretory Phospholipase A2 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50115782(1-(3-Trifluoromethyl-phenyl)-3-(2,4,6-trimethoxy-p...)
Affinity DataIC50:  1.84E+3nMAssay Description:Inhibitory concentration of the compound required to produce 50% inhibition of the response was determined; range-0.541.16 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50269844(CHEMBL517216 | Dysidine)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human synovial recombinant group 2 secretory phospholipase A2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50259951(CHEMBL480681 | cacospongionolide)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of bee venom group3 sPLA2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50259951(CHEMBL480681 | cacospongionolide)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of bee venom group3 sPLA2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50259951(CHEMBL480681 | cacospongionolide)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human synovial group2 sPLA2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcidic phospholipase A2 2(Naja naja)
Istituto Per La Chimica Di Molecole Di Interesse Biologico Cnr

Curated by ChEMBL
LigandPNGBDBM50259951(CHEMBL480681 | cacospongionolide)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Naja naja venom group1 sPLA2 at 10 uM by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-alkyl-2-acetylglycerophosphocholine esterase(Sus scrofa)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085496(CHEMBL89162 | N*1*,N*1*-Diethyl-hexadecane-1,2-dia...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of secretory PLA2 activity in porcine pancreas using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50259943((1R,3R,4aR,4bS,10aS,12aS)-3-(2-hydroxy-5-oxo-2,5-d...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human synovial secretory PLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50085497(2-(ethylamino)hexadecan-1-ol | 2-Ethylamino-hexade...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of secretory PLA2 activity in human recombinant synovial enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50259942(CHEMBL470340 | Petrosaspongiolide P)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human synovial secretory PLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibitory activity against human synovial recombinant Phospholipase enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of human synovial secretory PLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of human synovial group2 sPLA2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of human synovial recombinant group 2 secretory phospholipase A2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50066342(5-Hydroxy-4-[5-((2E,6E)-3,7,11-trimethyl-dodeca-2,...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibitory activity against human synovial recombinant Phospholipase enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50377908(CACOSPONGIONOLIDE B)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human synovial group2 sPLA2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50085496(CHEMBL89162 | N*1*,N*1*-Diethyl-hexadecane-1,2-dia...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of secretory PLA2 activity in human recombinant synovial enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50085497(2-(ethylamino)hexadecan-1-ol | 2-Ethylamino-hexade...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of secretory PLA2 activity in Naja naja venom enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50085497(2-(ethylamino)hexadecan-1-ol | 2-Ethylamino-hexade...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of secretory PLA2 activity in Naja naja venom enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibitory activity against bee secretory Phospholipase A2 enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of bee venom secretory PLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of bee venom group 3 secretory phospholipase A2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of bee venom group3 sPLA2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Rattus norvegicus)
Istituto Per La Chimica Di Molecole Di Interesse Biologico Cnr

Curated by ChEMBL
LigandPNGBDBM50259952(CHEMBL480874 | cacospongionolide E)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of rat air pouch group2 sPLA2 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50085496(CHEMBL89162 | N*1*,N*1*-Diethyl-hexadecane-1,2-dia...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of secretory PLA2 activity in bee venom enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Mus musculus)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085498(4-(1-Benzyloxymethyl-pentadecylcarbamoyl)-butyric ...)
Affinity DataIC50:  1.05E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50085496(CHEMBL89162 | N*1*,N*1*-Diethyl-hexadecane-1,2-dia...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of secretory PLA2 activity in bee venom enzyme using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Mus musculus)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085494(1,1,1-Trifluoro-heptadecan-2-oneor(Palmitoyl trifl...)
Affinity DataIC50:  1.17E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosolic phospholipase A2(Mus musculus)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085496(CHEMBL89162 | N*1*,N*1*-Diethyl-hexadecane-1,2-dia...)
Affinity DataIC50:  1.19E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcidic phospholipase A2 2(Naja naja)
Istituto Per La Chimica Di Molecole Di Interesse Biologico Cnr

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of Naja naja venom group1 sPLA2 at 10 uM by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Rattus norvegicus)
Istituto Per La Chimica Di Molecole Di Interesse Biologico Cnr

Curated by ChEMBL
LigandPNGBDBM50259951(CHEMBL480681 | cacospongionolide)
Affinity DataIC50:  2.18E+4nMAssay Description:Inhibition of rat air pouch group2 sPLA2 at 10 uM by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Apis mellifera)
Università

Curated by ChEMBL
LigandPNGBDBM50377908(CACOSPONGIONOLIDE B)
Affinity DataIC50:  3.54E+4nMAssay Description:Inhibition of bee venom group3 sPLA2 at 10 uM by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Rattus norvegicus)
Istituto Per La Chimica Di Molecole Di Interesse Biologico Cnr

Curated by ChEMBL
LigandPNGBDBM50377908(CACOSPONGIONOLIDE B)
Affinity DataIC50:  3.69E+4nMAssay Description:Inhibition of rat air pouch group2 sPLA2 at 10 uM by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Rattus norvegicus)
Istituto Per La Chimica Di Molecole Di Interesse Biologico Cnr

Curated by ChEMBL
LigandPNGBDBM50250399(5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...)
Affinity DataIC50:  3.84E+4nMAssay Description:Inhibition of rat air pouch group2 sPLA2 at 10 uM by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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