Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ki for monomerid = 50157672
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  22.3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  45.5nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  76.6nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  84.5nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed