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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50157672'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  84.5nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed