Affinity DataKi: 56nMAssay Description:In vitro binding affinity against rat histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 311nMAssay Description:Effect on specific [35S]-GTP-gammaS, Binding to HEK293 cell membranes expressing the human Histamine H3 receptorMore data for this Ligand-Target Pair