TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Stanford University
Curated by ChEMBL
Stanford University
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of mTOR kinase expressed in human HEK293 cells by western blot analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Stanford University
Curated by ChEMBL
Stanford University
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Inhibitory concentration against FKBP12 receptorMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Stanford University
Curated by ChEMBL
Stanford University
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:The inhibitory activity by using FK506 binding protein 12 SPA binding assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Stanford University
Curated by ChEMBL
Stanford University
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of mTOR (unknown origin) incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Stanford University
Curated by ChEMBL
Stanford University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mTOR-mediated Akt phosphorylation in human PC3 cellsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Stanford University
Curated by ChEMBL
Stanford University
Curated by ChEMBL
Affinity DataKd: 0.600nMAssay Description:Binding affinity to mTOR FKBP12 site (unknown origin)More data for this Ligand-Target Pair