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Found 7 Enz. Inhib. hit(s) with all data for entry = 50008953
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50078819(1-[4-((R)-3-Bromo-10-methoxy-8-methyl-6,11-dihydro...)
Affinity DataIC50:  3.60nMAssay Description:In vitro inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50078815(1-[4-(10-Methoxy-3,8-dimethyl-6,11-dihydro-5H-benz...)
Affinity DataIC50:  34nMAssay Description:In vitro inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50078814(1-[4-(10-Methoxy-8-methyl-3-vinyl-6,11-dihydro-5H-...)
Affinity DataIC50:  59nMAssay Description:In vitro inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50078818(1-[4-(3-Ethyl-10-methoxy-8-methyl-6,11-dihydro-5H-...)
Affinity DataIC50:  74nMAssay Description:In vitro inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50078817(1-[4-(10-Methoxy-8-methyl-6,11-dihydro-5H-benzo[5,...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50078816(1-[4-(3-Cyclopropyl-10-methoxy-8-methyl-6,11-dihyd...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM14459((+)-4-[2-[4-(8-Chloro-3,10-dibromo-6,11-dihydro-5H...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair