BDBM50078814 1-[4-(10-Methoxy-8-methyl-3-vinyl-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl)-piperidin-1-yl]-2-(1-oxy-pyridin-4-yl)-ethanone::CHEMBL56478

SMILES COc1cc(C)cc2CCc3cc(C=C)cnc3C(C3CCN(CC3)C(=O)Cc3cc[n+]([O-])cc3)c12

InChI Key InChIKey=XCDDGFBYFVYUQD-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50078814   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50078814(1-[4-(10-Methoxy-8-methyl-3-vinyl-6,11-dihydro-5H-...)
Affinity DataIC50:  59nMAssay Description:In vitro inhibition of human FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed