Compile Data Set for Download or QSAR
maximum 50k data
Found 34 Enz. Inhib. hit(s) with all data for entry = 50039143
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317250(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317246(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methy...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317253(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-iodo-N...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317248(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317251(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317254(CHEMBL1088507 | N-(azepan-1-yl)-1-(4-chlorophenyl)...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317252(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163112(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-ethy...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317245(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317255(CHEMBL1088376 | N-(azepan-1-yl)-5-(4-chlorophenyl)...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163122(1-(4-Chloro-phenyl)-5-cyano-2-(2,4-dichloro-phenyl...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163120(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317256(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(hydro...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50378776(1-(4-CHLOROPHENYL)-2-(2,4-DICHLOROPHENYL)-5-(METHY...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50378776(1-(4-CHLOROPHENYL)-2-(2,4-DICHLOROPHENYL)-5-(METHY...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317249(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(ethyl...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317254(CHEMBL1088507 | N-(azepan-1-yl)-1-(4-chlorophenyl)...)
Affinity DataKi:  325nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317255(CHEMBL1088376 | N-(azepan-1-yl)-5-(4-chlorophenyl)...)
Affinity DataKi:  371nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317245(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163112(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-ethy...)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163120(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  608nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317250(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  634nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317252(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  804nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317249(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(ethyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317246(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methy...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50378776(1-(4-CHLOROPHENYL)-2-(2,4-DICHLOROPHENYL)-5-(METHY...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50378776(1-(4-CHLOROPHENYL)-2-(2,4-DICHLOROPHENYL)-5-(METHY...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317251(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methy...)
Affinity DataKi:  1.07E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163122(1-(4-Chloro-phenyl)-5-cyano-2-(2,4-dichloro-phenyl...)
Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317253(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-iodo-N...)
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317256(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(hydro...)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50317248(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed