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Target
Somatostatin receptor type 5
Ligand
BDBM50370051
Substrate
n/a
Meas. Tech.
ChEMBL_200860 (CHEMBL807069)
Ki
176±n/a nM
Citation
 Rajeswaran, WG; Hocart, SJ; Murphy, WA; Taylor, JE; Coy, DH Highly potent and subtype selective ligands derived by N-methyl scan of a somatostatin antagonist. J Med Chem 44:1305-11 (2001) [PubMed]  Article 
Target
Name:
Somatostatin receptor type 5
Synonyms:
SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5)
Type:
Enzyme
Mol. Mass.:
39218.02
Organism:
Homo sapiens (Human)
Description:
P35346
Residue:
364
Sequence:
MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTLVIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDGVNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADVQEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRRRSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCANPVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQTSKL
  
Inhibitor
Name:
BDBM50370051
Synonyms:
CHEMBL1794043
Type:
Small organic molecule
Emp. Form.:
C60H71N13O9S2
Mol. Mass.:
1182.417
SMILES:
C[C@H](O)[C@H]1NC(=O)[C@H](CCCCN)N(C)C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)C(Cc2cccnc2)NC(=O)[C@H](CSSC[C@@H](NC1=O)C(=O)NC(Cc1c[nH]c2ccccc12)C(N)=O)NC(=O)C(N)Cc1ccc2ccccc2c1
Structure:
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