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Found 241 with Last Name = 'rajeswaran' and Initial = 'wg'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107697(1-[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107698(1,8-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107712(1,10-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  0.25nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107702(1,10-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107709(1,11-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107708(1,6-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  0.610nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107710(1,12-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl...)
Affinity DataKi:  0.690nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107696(1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  0.840nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107701(1,6-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  0.870nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107711(1,4-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  0.930nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107717(1,3-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  1.20nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-3 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  1.40nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107703(1-[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107715(1,12-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107713(1-[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  2nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-4 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370062(CHEMBL1794035)
Affinity DataKi:  2nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-1 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107716(1-[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)-1,2...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by displacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107704(1,8-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370053(CHEMBL1793861)
Affinity DataKi:  5.45nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370064(CHEMBL1794040)
Affinity DataKi:  5.98nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107699(1,7-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  7.60nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370057(CHEMBL1794039)
Affinity DataKi:  9.33nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50098908(CHEMBL262899 | Tfm-cyclo(DCys-Pal-DTrp-NMeLys-Thr-...)
Affinity DataKi:  11.3nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370050(CHEMBL1794032)
Affinity DataKi:  12.1nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107706(1,5-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  14nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107705(1,9-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  17nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370064(CHEMBL1794040)
Affinity DataKi:  17.1nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107707(1,2-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl)...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370066(CHEMBL1794045)
Affinity DataKi:  23.6nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-3 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370048(CHEMBL1794042)
Affinity DataKi:  24.7nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370051(CHEMBL1794043)
Affinity DataKi:  27.3nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370058(CHEMBL1794033)
Affinity DataKi:  36nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370050(CHEMBL1794032)
Affinity DataKi:  38.2nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-3 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370058(CHEMBL1794033)
Affinity DataKi:  40.1nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50098908(CHEMBL262899 | Tfm-cyclo(DCys-Pal-DTrp-NMeLys-Thr-...)
Affinity DataKi:  40.2nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-3 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50098908(CHEMBL262899 | Tfm-cyclo(DCys-Pal-DTrp-NMeLys-Thr-...)
Affinity DataKi:  45.5nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370060(CHEMBL1794036)
Affinity DataKi:  51.8nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370064(CHEMBL1794040)
Affinity DataKi:  66nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-3 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370055(CHEMBL1793860)
Affinity DataKi:  68.7nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-3 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)
Affinity DataKi:  82nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370061(CHEMBL1794037)
Affinity DataKi:  88.5nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370056(CHEMBL1794034)
Affinity DataKi:  89nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-2 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370053(CHEMBL1793861)
Affinity DataKi:  91.4nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-3 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370060(CHEMBL1794036)
Affinity DataKi:  93nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370053(CHEMBL1793861)
Affinity DataKi:  101nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370056(CHEMBL1794034)
Affinity DataKi:  106nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Tulane University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50370057(CHEMBL1794039)
Affinity DataKi:  112nMAssay Description:Ability to displace [125 I]labelled Tyr11-somatostatin from human hsst-5 receptor expressed on CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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