BDBM135616 US10179804, Example 1::US10632171, Peptide No. 1::US8846601, 1::US8846601, 115::US8846601, 51::US9458201, 115

SMILES CC(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@H]1CC(=O)NCCCC[C@H](NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]cn2)NC1=O)C(N)=O

InChI Key

Data  8 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 135616   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135616(US10179804, Example 1 | US10632171, Peptide No. 1 ...)
Affinity DataKi:  5nM ΔG°:  -11.8kcal/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135616(US10179804, Example 1 | US10632171, Peptide No. 1 ...)
Affinity DataKi:  22nM ΔG°:  -10.9kcal/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135616(US10179804, Example 1 | US10632171, Peptide No. 1 ...)
Affinity DataKi:  87nM ΔG°:  -10.0kcal/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent