BDBM14525 N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-3-(methylamino)-2-oxo-6-phenyl-1,2-dihydropyrazin-1-yl]acetamide::Pyrazinone Analog 28a
SMILES CNc1nc(Cl)c(-c2ccccc2)n(CC(=O)NCc2ccc(cc2)C(N)=N)c1=O
InChI Key InChIKey=GHNPQZVQEKZFKF-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 14525
Affinity DataIC50: 700nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+4nMAssay Description:Human thrombin and substrate were added to a 96-well assay plate containing inhibitor in reaction buffer. The rate of hydrolysis of the substrate was...More data for this Ligand-Target Pair