BDBM14542 N-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-3-(cyclobutylamino)-2-oxo-6-phenyl-1,2-dihydropyrazin-1-yl]acetamide::Pyrazinone Analog 28m
SMILES NC(=N)c1ccc(CNC(=O)Cn2c(c(Cl)nc(NC3CCC3)c2=O)-c2ccccc2)cc1
InChI Key InChIKey=VZWRMPXNNHXNHC-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 14542
Affinity DataIC50: 400nMAssay Description:Recombinant human Factor VIIa and soluble tissue factor were added to a 96-well assay plate containing substrate and inhibitor in reaction buffer. Th...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Human thrombin and substrate were added to a 96-well assay plate containing inhibitor in reaction buffer. The rate of hydrolysis of the substrate was...More data for this Ligand-Target Pair