BDBM18573 6-(cyclopentylamino)-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one::6-alkylamino 2-quinolinone, 13e

SMILES FC(F)(F)c1cc(=O)[nH]c2ccc(NC3CCCC3)cc12

InChI Key InChIKey=WUSYUUHWBCIJBB-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 18573   

TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

LigandPNGBDBM18573(6-(cyclopentylamino)-4-(trifluoromethyl)-1,2-dihyd...)
Affinity DataKi:  74nM IC50:  42nMAssay Description:The compounds were evaluated in a transcriptional activation assay with hAR in a mammalian cell background (CV-1) as the primary in vitro assay. Rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed