BDBM195753 US9206173, 166
SMILES C[C@@H](Nc1nc2CCN(Cc2c(=O)n1N1CCCC1)C(=O)c1ccc(cc1F)C#N)c1ccc(cc1)C(F)(F)F
InChI Key InChIKey=UKUPQDJSUUDRIY-QGZVFWFLSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 195753
Affinity DataKi: 6nM ΔG°: -11.2kcal/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
Affinity DataIC50: 298nMpH: 7.4 T: 2°CAssay Description:HEK293 cells expressing human GPR10 were maintained in Dulbecco's Modified Eagles' medium supplemented with 10% fetal bovine serum, 1% penici...More data for this Ligand-Target Pair