BDBM196909 US9212196, Derivative 5

SMILES COc1cc(cc(c1OCC(O)=O)[N+]([O-])=O)C(O)P(O)(=O)CC[C@@H](N)C(O)=O

InChI Key InChIKey=OCWGTIQPGGIBEM-ZSYIFEHUSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 196909   

TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Universite Paris Descartes

US Patent
LigandPNGBDBM196909(US9212196, Derivative 5)
Affinity DataEC50:  280nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Universite Paris Descartes

US Patent
LigandPNGBDBM196909(US9212196, Derivative 5)
Affinity DataEC50: >1.00E+5nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Universite Paris Descartes

US Patent
LigandPNGBDBM196909(US9212196, Derivative 5)
Affinity DataEC50:  5.95E+3nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Universite Paris Descartes

US Patent
LigandPNGBDBM196909(US9212196, Derivative 5)
Affinity DataEC50:  3.72E+3nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent