BDBM200870 US9533999, i-23

SMILES Fc1ccc(CN2C(=O)CS(=O)(=O)c3nccnc23)cc1OC(F)(F)F

InChI Key InChIKey=CEMONOUPMAZYPE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 200870   

TargetIntermediate conductance calcium-activated potassium channel protein 4(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM200870(US9533999, i-23)
Affinity DataIC50:  170nMAssay Description:HEK293 cells over-expressing human KCa3.1 are used to measure the effects of compounds in inhibiting the KCa3.1 channel function. The assay is based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent