BDBM20196 3, Ac-pTyr-Leu-Pro-Gln-NH2::4-[(2S)-2-{[(2S)-1-[(2S)-2-{[(1S)-1,3-dicarbamoylpropyl]carbamoyl}pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid::BMCL13633 gp130 (904) derived peptide, 18::CHEMBL194516

SMILES CC(C)C[C@H](NC(=O)[C@H](Cc1ccc(OP(O)(O)=O)cc1)NC(C)=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(N)=O)C(N)=O

InChI Key InChIKey=VRWGJYWTUFHEQV-CMOCDZPBSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 20196   

TargetSignal transducer and activator of transcription 3(Mus musculus (mouse))
The University of Texas At Houston

LigandPNGBDBM20196(3, Ac-pTyr-Leu-Pro-Gln-NH2 | 4-[(2S)-2-{[(2S)-1-[(...)
Affinity DataIC50:  856nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization (FP) binding assay is utilizing the intrinsic property of the fluorescent probe, which will have low polarization value whe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM20196(3, Ac-pTyr-Leu-Pro-Gln-NH2 | 4-[(2S)-2-{[(2S)-1-[(...)
Affinity DataIC50:  856nMAssay Description:Inhibition of Stat3 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Mus musculus (mouse))
The University of Texas At Houston

LigandPNGBDBM20196(3, Ac-pTyr-Leu-Pro-Gln-NH2 | 4-[(2S)-2-{[(2S)-1-[(...)
Affinity DataIC50:  1.00E+3nMpH: 7.8 T: 2°CAssay Description:His10-Stat3 was expressed in Sf9 cells from a baculovirus encoding the recombinant protein. A nuclear extract of the Sf9 cells was incubated with 32P...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed