BDBM23029 1-[5-(pyridin-2-yl)-1,3-oxazol-2-yl]-7-(thiophen-3-yl)heptan-1-one::alpha-ketooxazole, 5b
SMILES O=C(CCCCCCc1ccsc1)c1ncc(o1)-c1ccccn1
InChI Key InChIKey=BBFQYOOSPUJNBB-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 23029
Affinity DataKi: 5.10nM ΔG°: -11.2kcal/mole IC50: 40nMpH: 9.0 T: 2°CAssay Description:The inhibition assays were performed by incubating enzyme, 14C-labeled oleamide in reaction buffer at room temperature in the presence of three diffe...More data for this Ligand-Target Pair
Affinity DataIC50: 800nMT: 2°CAssay Description:Inhibition of TGH activity was assayed using COS-7 expressed TGH and the chromogenic substrate. IC50 values were determined from the inhibition obser...More data for this Ligand-Target Pair