BDBM241188 US11046688, Example 30::US9409907, 30
SMILES COc1ccc(Nc2cc3c(cccc3cn2)-c2cnn(C)c2)c(OC)c1
InChI Key InChIKey=SEROCBXXHACDIM-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 241188
Affinity DataIC50: 74nMpH: 7.0 T: 2°CAssay Description:The enzyme reaction (total volume 10 μl) was carried out in black 384-well low volume plates containing full length MPS1 (12.5 nM or 3 nM), fluo...More data for this Ligand-Target Pair