BDBM243059 PTP inhibitor, 4k
SMILES Oc1cc(O)c2C(=O)CC(Oc2c1)c1cccc(c1)C(F)(F)F
InChI Key InChIKey=JPSPQWKZLGZAHP-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 243059
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Yanbian University College of Pharmacy
Yanbian University College of Pharmacy
Affinity DataIC50: 2.37E+3nMpH: 6.5 T: 2°CAssay Description:Briefly, the enzymatic activity of the PTP1B catalytic domain was determinedat 30°C by monitoring the hydrolysis of pNPP. Dephosphorylation of pNPP g...More data for this Ligand-Target Pair
Affinity DataIC50: 8.54E+3nMpH: 6.5 T: 2°CAssay Description:Briefly, the enzymatic activity of the PTP1B catalytic domain was determinedat 30°C by monitoring the hydrolysis of pNPP. Dephosphorylation of pNPP g...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Yanbian University College of Pharmacy
Yanbian University College of Pharmacy
Affinity DataIC50: 8.82E+3nMpH: 6.5 T: 2°CAssay Description:Briefly, the enzymatic activity of the PTP1B catalytic domain was determinedat 30°C by monitoring the hydrolysis of pNPP. Dephosphorylation of pNPP g...More data for this Ligand-Target Pair