BDBM270918 4-cyclohexyl-7-{[4-(difluoromethoxy)benzene]sulfonyl}-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 36
SMILES Nc1[nH]c2c(ncnc2c1S(=O)(=O)c1ccc(OC(F)F)cc1)C1CCCCC1
InChI Key InChIKey=ZWOOWQAMLSSBIO-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 270918
Affinity DataEC50: 87nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair