BDBM283255 US10023543, Example 40::US10207999, Example 40::US10328077, Example 40::US10548896, Example 40::US10849898, Example 40::US10960005, Example 40::US11084793, Example 40::US9573930, Example 40::US9771329, Example 40::US9776974, Example 40::{4-[2-(4-aminopiperidyl)-6- (4-cyanophenyl)-3-methyl-4-oxo (3-hydro pyrimidin-5-yl)]-2- fluorophenyl}-N- methylcarboxamide
SMILES CNC(=O)c1ccc(cc1F)-c1c(nc(N2CCC(N)CC2)n(C)c1=O)-c1ccc(cc1)C#N
InChI Key InChIKey=JRYTXSJOBAOEPP-UHFFFAOYSA-N
Data 12 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 283255
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Celgene Quanticel Research
US Patent
Affinity DataIC50: <100nMT: 2°CAssay Description:This assay determines the ability of a test compound to inhibit LSD1 demethylase activity. E. coli expressed full-length human LSD1 (Accession number...More data for this Ligand-Target Pair