BDBM286722 N-{(R)-1-[6-Bromo-3-(5-chloro-2-ethanesulfonyl-benzyl)-2,4-dioxo-1,2,3,4-tetrahydro-quinazolin-7-ylmethyl]-pyrrolidin-3-yl}-dimethylaminosulfonamide::US9567304, Compound E-10

SMILES CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NS(=O)(=O)N(C)C)c(Br)cc2c1=O

InChI Key InChIKey=PTQDOTHLLUMOST-GOSISDBHSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 286722   

TargetEpithelial discoidin domain-containing receptor 1(Homo sapiens (Human))
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandPNGBDBM286722(N-{(R)-1-[6-Bromo-3-(5-chloro-2-ethanesulfonyl-ben...)
Affinity DataIC50:  15nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent