BDBM28676 5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoquinoline-2-)sulfonyl]benzene}amido)benzoic acid::Anthranilic acid deriv., 15

SMILES COc1ccc2CN(CCc2c1)S(=O)(=O)c1cccc(c1)C(=O)Nc1ccc(Cl)cc1C(O)=O

InChI Key InChIKey=FYIPIRTZBJMPOQ-UHFFFAOYSA-N

Data  9 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 28676   

LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  10nM EC50:  794nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  1.00E+4nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  6.31E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  1.00E+4nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  6.31E+3nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  6.31E+3nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  1.00E+4nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  10nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28676(5-chloro-2-({3-[(6-methoxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataIC50:  10nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed