BDBM34144 (R)-5a::WAY-466

SMILES [H][C@]1(Cc2c[nH]c3ccc(NS(=O)(=O)c4ccccc4I)cc23)CCCN1

InChI Key InChIKey=ZLTKHJVPOSETMR-CQSZACIVSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 34144   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universitat De Barcelona

LigandPNGBDBM34144((R)-5a | WAY-466)
Affinity DataKi:  1nM ΔG°:  -12.8kcal/mole EC50:  0.400nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed